Search on: LACTATE, PENTAZOCINE 
Descriptors Found: 1
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Descriptor English:   Pentazocine 
Descriptor Spanish:   Pentazocina 
Descriptor Portuguese:   Pentazocina 
Synonyms English:   Fortral
Lexir
Pentazocine Hydrochloride
Pentazocine Lactate
Talwin
Hydrochloride, Pentazocine
Lactate, Pentazocine  
Tree Number:   D03.132.577.249.106.700
D04.615.723.795.106.700
Definition English:   The first mixed agonist-antagonist analgesic to be marketed. It is an agonist at the kappa and sigma opioid receptors and has a weak antagonist action at the mu receptor. (From AMA Drug Evaluations Annual, 1991, p97) 
Pharmacological Action:   Adjuvants, Anesthesia
Analgesics, Opioid
Narcotic Antagonists
Narcotics
 
History Note English:   66(64) 
Allowable Qualifiers English:  
AD administration & dosage AE adverse effects
AG agonists AA analogs & derivatives
AN analysis AI antagonists & inhibitors
BL blood CF cerebrospinal fluid
CS chemical synthesis CH chemistry
CL classification CT contraindications
EC economics HI history
IM immunology IP isolation & purification
ME metabolism PK pharmacokinetics
PD pharmacology PO poisoning
RE radiation effects ST standards
SD supply & distribution TU therapeutic use
TO toxicity UR urine
Record Number:   10617 
Unique Identifier:   D010423 

Occurrence in VHL:
 

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